Bisnortilidine
Appearance
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Preferred IUPAC name
Ethyl (1R,2S)-2-amino[1,1′-bi(cyclohexane)]-1′,3,3′,5′-tetraene-1-carboxylate | |
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3D model (JSmol)
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Properties | |
C15H19NO2 | |
Molar mass | 245.322 g·mol−1 |
Except where otherwise noted, data are given for materials in their standard state (at 25 °C [77 °F], 100 kPa).
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Bisnortilidine is an opioid metabolite.[1] It is formed from tilidine by demethylation in the liver.
References
[edit]- ^ Wustrow, I.; Riedel, K. D.; Mikus, G.; Weiss, J. (2012). "In vitro identification of the cytochrome P450 isozymes involved in the N-demethylation of the active opioid metabolite nortilidine to bisnortilidine". Naunyn-Schmiedeberg's Archives of Pharmacology. 385 (6): 633–9. doi:10.1007/s00210-012-0737-z. PMID 22349139. S2CID 2660215.